All

What are you looking for?

All
Projects
Results
Organizations

Quick search

  • Projects supported by TA ČR
  • Excellent projects
  • Projects with the highest public support
  • Current projects

Smart search

  • That is how I find a specific +word
  • That is how I leave the -word out of the results
  • “That is how I can find the whole phrase”

Fused Ring Molecular Scaffold with 3D Architecture for Constrained Peptidomimetics: Polymer-Supported Stereoselective Synthesis of Tetrahydrobenzo[e]pyrazinothiadiazinone 6,6-dioxide via N-Acyl Iminiums

The result's identifiers

  • Result code in IS VaVaI

    <a href="https://www.isvavai.cz/riv?ss=detail&h=RIV%2F61989592%3A15110%2F16%3A33160874" target="_blank" >RIV/61989592:15110/16:33160874 - isvavai.cz</a>

  • Result on the web

    <a href="http://pubs.acs.org/doi/ipdf/10.1021/acscombsci.6b00126" target="_blank" >http://pubs.acs.org/doi/ipdf/10.1021/acscombsci.6b00126</a>

  • DOI - Digital Object Identifier

    <a href="http://dx.doi.org/10.1021/acscombsci.6b00126" target="_blank" >10.1021/acscombsci.6b00126</a>

Alternative languages

  • Result language

    angličtina

  • Original language name

    Fused Ring Molecular Scaffold with 3D Architecture for Constrained Peptidomimetics: Polymer-Supported Stereoselective Synthesis of Tetrahydrobenzo[e]pyrazinothiadiazinone 6,6-dioxide via N-Acyl Iminiums

  • Original language description

    3,4,4a,5-Tetrahydrobenzo[e]pyrazinothiadiazin-1(2H)-one 6,6-dioxides, molecular scaffolds with 3D architecture, were synthesized on a solid support via tandem N-acyl iminium ion cyclization followed by nucleophilic addition. The modular synthesis proceeded under mild conditions using commercially available building blocks and provided crude products with respectable purity. Synthesized compounds are applicable as fused nitrogenous heterocyclic compounds in drug discovery as well as constrained peptidomimetics incorporated into peptide backbone.

  • Czech name

  • Czech description

Classification

  • Type

    J<sub>x</sub> - Unclassified - Peer-reviewed scientific article (Jimp, Jsc and Jost)

  • CEP classification

    CC - Organic chemistry

  • OECD FORD branch

Result continuities

  • Project

    Result was created during the realization of more than one project. More information in the Projects tab.

  • Continuities

    P - Projekt vyzkumu a vyvoje financovany z verejnych zdroju (s odkazem do CEP)

Others

  • Publication year

    2016

  • Confidentiality

    S - Úplné a pravdivé údaje o projektu nepodléhají ochraně podle zvláštních právních předpisů

Data specific for result type

  • Name of the periodical

    ACS Combinatorial Science

  • ISSN

    2156-8952

  • e-ISSN

  • Volume of the periodical

    18

  • Issue of the periodical within the volume

    10

  • Country of publishing house

    US - UNITED STATES

  • Number of pages

    5

  • Pages from-to

    655-659

  • UT code for WoS article

  • EID of the result in the Scopus database