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475 (0,063s)

Result

Identification and Validation of Compounds Targeting Leishmania major Leucyl-Aminopeptidase M17

is M17 leucyl-aminopeptidase (LAP). Here, we aimed to chemically validate LAP. Thermal proteome profiling revealed that these inhibitors thermally stabilized two M17......

Cell biology

  • 2024
  • Jimp
  • Link
Result

Identification of a potent and selective LAPTc inhibitor by RapidFire-Mass Spectrometry, with antichagasic activity

are urgently required. Here we identified inhibitors of the acidic M17 leucyl-aminopeptidase from T. cruzi (LAPTc) that show promise as novel starting points for Chagas......

Infectious Diseases

  • 2024
  • Jimp
  • Link
Result

Isozymes of phosphatase and leucine and leucine aminopeptidase as biochemical markers for purity testing in rapeseed androgenetic lines.m

EB - Genetika a molekulární biologie

  • 1994
  • Jx
Result

Identification and Validation of Compounds Targeting Leishmania major Leucyl-Aminopeptidase M17

is M17 leucyl-aminopeptidase (LAP). Here, we aimed to chemically validate LAP. Thermal proteome profiling revealed that these inhibitors thermally stabilized two M17......

Cell biology

  • 2024
  • Jimp
  • Link
Result

A leucine aminopeptidase is involved in kinetoplast DNA segregation in Trypanosoma brucei

the daughter kDNA networks prior to their segregation. Here we characterize an M17 family leucyl aminopeptidase metalloprotease, termed TbLAP1, which specifically localizes......

Biochemistry and molecular biology

  • 2017
  • Jimp
  • Link
Result

A leucine aminopeptidase is involved in kinetoplast DNA segregation in Trypanosoma brucei

the daughter kDNA networks prior to their segregation. Here we characterize an M17 family leucyl aminopeptidase metalloprotease, termed TbLAP1, which specifically localizes......

Genetics and heredity (medical genetics to be 3)

  • 2017
  • Jimp
  • Link
Result

Development of a High-Throughput Screening Assay to Identify Inhibitors of the Major M17-Leucyl Aminopeptidase from Trypanosoma cruzi Using RapidFire Mass Spectrometry

Leucyl aminopeptidases (LAPs) are involved in multiple cellular functions, which, in the case of infectious diseases, includes participation in the pathogen-host cell interface and pathogenesis. Thus, LAPs are considered good candidate drug ...

Biological sciences

  • 2020
  • Jimp
  • Link
Result

Unusual activity pattern of leucine aminopeptidase inhibitors based on phosphorus containing derivatives of methionine and norleucine

Ligands containing bulky aliphatic P1 residues exhibit a high affinity towards cytosolic leucine aminopeptidase, a bizinc protease of biomedical significance. According to this specificity, a series of phosphonic and phosphinic comp...

CC - Organická chemie

  • 2011
  • Jx
  • Link
Result

Acid phosphatase and leucine aminopeptidase isozymes as biochemical markers of homogenity in oil seed rape androgenetic lines

EB - Genetika a molekulární biologie

  • 1994
  • Jx
Result

Acid phosphatase and leucine aminopeptidase isozymes as biochemical markers of homogenity in oil seed rape androgenetic linies

EB - Genetika a molekulární biologie

  • 1995
  • Jx
  • 1 - 10 out of 475