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168 738 (0,152s)

Result

Ligand-Based Pharmacophore Modeling Using Novel 3D Pharmacophore Signatures

Pharmacophore modeling is a widely used strategy for finding new hit molecules, a 3D pharmacophore ligand-based modeling approach to search for pharmacophores. The approach searches for 3D pharmacophor...

Biochemistry and molecular biology

  • 2018
  • Jimp
  • Link
Result

2D Pharmacophore Query Generation

and compiled into a 3D pharmacophore model. However, in many cases the structures of the ligands are not known which results in using a 2D pharmacophore model. We introduce a method capable of automatic generation...

IN - Informatika

  • 2014
  • D
  • Link
Result

Probabilistic Approach for Virtual Screening Based on Multiple Pharmacophores

Pharmacophore modeling is a widely used approach for the discovery of new biologically active compounds. According to the IUPAC definition, pharmacophore of successful applications of pharmacophore models ...

Biochemistry and molecular biology

  • 2020
  • Jimp
  • Link
Result

Comprehensive Comparison of the Ergot Alkaloids Family with 5-HT Receptor Pharmacophore Models

Comprehensive Comparison of the Ergot Alkaloids Family with 5_HT Receptor Pharmacophore Models...

CC - Organická chemie

  • 2000
  • A
Result

Comprehensive Comparison of the Ergot Alkaloids Family with 5 -HT Receptor Pharmacophore Models.

Comprehensive Comparison of the Ergot Alkaloids Family with 5-HT Receptor Pharmacophore Models...

CC - Organická chemie

  • 2000
  • D
Result

Pharmacophore Modelling Used in Rational Drug Design

and is mainly focused on pharmacophore modelling, one of the modern approaches in drug...

Organic chemistry

  • 2016
  • Jimp
  • Link
Result

Use of 3D QSAR Pharmacophore Modelling in the Research of Influenza

, higher safety and increased tolerability. A pharmacophore is a set of structural at a receptor site and its biological activity. In the current work, 3D pharmacophore based pharmacophoric features present in the active s...

Biochemistry and molecular biology

  • 2016
  • D
  • Link
Result

In silico pharmacophore modeling on known pyridinium oxime reactivators of cyclosarin (GF) inhibited AChE to aid discovery of potential, more efficacious novel non-oxime reactivators

of novel antidotes for GF toxicity, a three-dimensional in silico pharmacophore model for reactivation efficacy against GF intoxication is presented. The model was generated from. The generated pharmacophore m...

FR - Farmakologie a lékárnická chemie

  • 2013
  • Jx
  • Link
Result

Antimycobacterial activita of compounds with basic pharmacophore. Piperidinoesters of phenylcarbamoyl acid.

New basic pharmacophore of antimycobacterial activity...

CC - Organická chemie

  • 2001
  • Jx
Result

Calculations of Resonance substituent Constatnts of some Important Pharmacophore Groups

Calculations of Resonance Substituent Constatnts of some Important Pharmacophore Groups...

CC - Organická chemie

  • 2001
  • D
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