All

What are you looking for?

All
Projects
Results
Organizations

Quick search

  • Projects supported by TA ČR
  • Excellent projects
  • Projects with the highest public support
  • Current projects

Smart search

  • That is how I find a specific +word
  • That is how I leave the -word out of the results
  • “That is how I can find the whole phrase”

Helquat derivatives, preparation thereof, and use thereof as medicaments

The result's identifiers

  • Result code in IS VaVaI

    <a href="https://www.isvavai.cz/riv?ss=detail&h=RIV%2F61388963%3A_____%2F16%3A00471681" target="_blank" >RIV/61388963:_____/16:00471681 - isvavai.cz</a>

  • Result on the web

    <a href="https://worldwide.espacenet.com/publicationDetails/biblio?CC=US&NR=9340543B2&KC=B2&FT=D&ND=4&date=20160517&DB=&locale=en_EP" target="_blank" >https://worldwide.espacenet.com/publicationDetails/biblio?CC=US&NR=9340543B2&KC=B2&FT=D&ND=4&date=20160517&DB=&locale=en_EP</a>

  • DOI - Digital Object Identifier

Alternative languages

  • Result language

    angličtina

  • Original language name

    Helquat derivatives, preparation thereof, and use thereof as medicaments

  • Original language description

    The invention provides helquat derivatives of general formula I, wherein substituents R1 and R2 are independently selected from a group comprising H and C1 to C3 alkyl; up to three of S1,2, S1',2', S3,4 and S3', 4' are present, each of S1,2, S1',2', S3,4 and S3',4' independently represents a linker consisting of a bivalent hydrocarbon chain having 3-6 carbon atoms; one or two atoms selected from the carbon atoms with the descriptor 2, 4, 2', and 4' are substituted with a substituent R3 of general formula II or general formula III wherein R4 is substituted or unsubstituted aryl; T1 and T2 independently represent a bivalent hydrocarbon chain having 2-5 carbon atoms; and anions (X1)- and (X2)- independently represent anions of pharmaceutically acceptable salts. The helquat derivatives are useful as medicaments in the treatment of diseases related to increased cellular proliferation, such as oncologic diseases.

  • Czech name

  • Czech description

Classification

  • Type

    P - Patent

  • CEP classification

    CC - Organic chemistry

  • OECD FORD branch

Result continuities

  • Project

  • Continuities

    I - Institucionalni podpora na dlouhodoby koncepcni rozvoj vyzkumne organizace

Others

  • Publication year

    2016

  • Confidentiality

    S - Úplné a pravdivé údaje o projektu nepodléhají ochraně podle zvláštních právních předpisů

Data specific for result type

  • Patent/design ID

    US9340543

  • Publisher

    US001 -

  • Publisher name

    United States Patent and Trademark Office (USPTO)

  • Place of publication

    Alexandria

  • Publication country

    US - UNITED STATES

  • Date of acceptance

    May 17, 2016

  • Owner name

    Ústav organické chemie a biochemie AV ČR, v. v. i

  • Method of use

    A - Výsledek využívá pouze poskytovatel

  • Usage type

    A - K využití výsledku jiným subjektem je vždy nutné nabytí licence