Solid-Phase Synthesis of Trisubstituted 2,5-Dihydrobenzo[f]thiadiazepine 1,1-Dioxide Derivatives

Result code in IS VaVaI
<a href="https://www.isvavai.cz/riv?ss=detail&h=RIV%2F61989592%3A15310%2F14%3A33151963" target="_blank" >RIV/61989592:15310/14:33151963 - isvavai.cz</a>
Result on the web
<a href="http://pubs.acs.org/doi/pdf/10.1021/co500084k" target="_blank" >http://pubs.acs.org/doi/pdf/10.1021/co500084k</a>
DOI - Digital Object Identifier
<a href="http://dx.doi.org/10.1021/co500084k" target="_blank" >10.1021/co500084k</a>

Result language
angličtina
Original language name
Solid-Phase Synthesis of Trisubstituted 2,5-Dihydrobenzo[f]thiadiazepine 1,1-Dioxide Derivatives
Original language description
The solid-phase synthesis of trisubstituted 2,5-dihydrobenzo[f]thiadiazepine 1,1-dioxides is reported. Acyclic polymer-supported intermediates were prepared using commercially available building blocks: Fmoc-protected amino acids, 2-nitrobenzenesulfonylchlorides, and bromoketones. The acyclic precursors underwent acid-mediated release from the resin and the cyclization was completed in solution.
Czech name
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Czech description
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Type
J<sub>x</sub> - Unclassified - Peer-reviewed scientific article (Jimp, Jsc and Jost)
CEP classification
CC - Organic chemistry
OECD FORD branch
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Project
Result was created during the realization of more than one project. More information in the Projects tab.
Continuities
P - Projekt vyzkumu a vyvoje financovany z verejnych zdroju (s odkazem do CEP)

Publication year
2014
Confidentiality
S - Úplné a pravdivé údaje o projektu nepodléhají ochraně podle zvláštních právních předpisů

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